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Impact of Renal Impairment on the Pharmacokinetics of Apremilast and Metabolite M12

The pharmacokinetics of apremilast and its major metabolite M12 were evaluated in subjects with varying degrees of renal impairment. Men and women with renal impairment (estimated glomerular filtration rate, 60‒89 mL/min [mild, n = 8], 30‒59 mL/min [moderate, n = 8], or <30 mL/min [severe, n = 8]...

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Publicat a:Clin Pharmacol Drug Dev
Autors principals: Liu, Yong, Zhou, Simon, Assaf, Mahmoud, Nissel, Jim, Palmisano, Maria
Format: Artigo
Idioma:Inglês
Publicat: John Wiley and Sons Inc. 2016
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5132082/
https://ncbi.nlm.nih.gov/pubmed/27870479
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cpdd.256
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