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Mechanism of Enhanced Cellular Uptake and Cytosolic Retention of MK2 Inhibitory Peptide Nano-polyplexes

Electrostatic complexation of a cationic MAPKAP kinase 2 inhibitory (MK2i) peptide with the anionic, pH-responsive polymer poly(propylacrylic acid) (PPAA) yields MK2i nano-polyplexes (MK2i-NPs) that significantly increase peptide uptake and intracellular retention. This study focused on elucidating...

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Publicado en:Cell Mol Bioeng
Autores principales: Kilchrist, Kameron V, Evans, Brian C, Brophy, Colleen M, Duvall, Craig L.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2016
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC5089375/
https://ncbi.nlm.nih.gov/pubmed/27818713
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s12195-016-0446-7
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