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In vitro metabolism of piperaquine is primarily mediated by CYP3A4
1. Piperaquine (PQ) is part of a first-line treatment regimen for Plasmodium falciparum malaria recommended by the World Health Organization (WHO). We aimed to determine the major metabolic pathway(s) of PQ in vitro. A reliable, validated tandem mass spectrometry method was developed. Concentrations...
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| Publicat a: | Xenobiotica |
|---|---|
| Autors principals: | , , , , , , |
| Format: | Artigo |
| Idioma: | Inglês |
| Publicat: |
2012
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| Matèries: | |
| Accés en línia: | https://ncbi.nlm.nih.gov/pmc/articles/PMC5087332/ https://ncbi.nlm.nih.gov/pubmed/22671777 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3109/00498254.2012.693972 |
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