Characterization of SR 121463A, a highly potent and selective, orally active vasopressin V2 receptor antagonist.

SR 121463A, a potent and selective, orally active, nonpeptide vasopressin V2 receptor antagonist, has been characterized in several in vitro and in vivo models. This compound displayed highly competitive and selective affinity for V2 receptors in rat, bovine and human kidney (0.6 < or = Ki [nM] &...

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Autores principales: Serradeil-Le Gal, C, Lacour, C, Valette, G, Garcia, G, Foulon, L, Galindo, G, Bankir, L, Pouzet, B, Guillon, G, Barberis, C, Chicot, D, Jard, S, Vilain, P, Garcia, C, Marty, E, Raufaste, D, Brossard, G, Nisato, D, Maffrand, J P, Le Fur, G
Formato: Artigo
Lenguaje:Inglês
Publicado: 1996
Materias:
Research Article
Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC507737/
https://ncbi.nlm.nih.gov/pubmed/8981918
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