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Identification and Characterization of CINPA1 Metabolites Facilitates Structure-Activity Studies of the Constitutive Androstane Receptor

The constitutive androstane receptor (CAR) regulates the expression of genes involved in drug metabolism and other processes. A specific inhibitor of CAR is critical for modulating constitutive CAR activity. We recently described a specific small-molecule inhibitor of CAR, CINPA1 (ethyl (5-(diethylg...

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Detalles Bibliográficos
Publicado en:Drug Metab Dispos
Main Authors: Cherian, Milu T., Yang, Lei, Chai, Sergio C., Lin, Wenwei, Chen, Taosheng
Formato: Artigo
Idioma:Inglês
Publicado: The American Society for Pharmacology and Experimental Therapeutics 2016
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC5074473/
https://ncbi.nlm.nih.gov/pubmed/27519550
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.116.071993
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