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Discovery of Novel Potent and Selective Agonists at the Melanocortin-3 Receptor

The melanocortin receptors 3 and 4 control energy homeostasis, food-intake behavior, and correlated pathophysiological conditions. The melanocortin-4 receptor (MC4R) has been broadly investigated. In contrast, the knowledge related to physiological roles of the melanocortin-3 receptor (MC3R) is lack...

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Publicado en:J Med Chem
Autores principales: Carotenuto, Alfonso, Merlino, Francesco, Cai, Minying, Brancaccio, Diego, Yousif, Ali Munaim, Novellino, Ettore, Hruby, Victor J., Grieco, Paolo
Formato: Artigo
Lenguaje:Inglês
Publicado: 2015
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC5070805/
https://ncbi.nlm.nih.gov/pubmed/26599352
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.5b01285
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