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Conformational study on cyclic melanocortin ligands and new insight into their binding mode at the MC4 receptor

The melanocortin receptors are involved in many physiological functions, including pigmentation, sexual function, feeding behavior, and energy homeostasis, making them potential targets to treat obesity, sexual dysfunction, etc. Understanding the basis of the ligand-receptor interactions is crucial...

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Detalles Bibliográficos
Publicado en:Eur J Med Chem
Autores principales: Grieco, Paolo, Brancaccio, Diego, Novellino, Ettore, Hruby, Victor J., Carotenuto, Alfonso
Formato: Artigo
Lenguaje:Inglês
Publicado: 2011
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC5102844/
https://ncbi.nlm.nih.gov/pubmed/21652123
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ejmech.2011.05.038
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