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Synthesis and pharmacological evaluation of indole derivatives as deaza analogues of potent human neutrophil elastase inhibitors (HNE)

A number of N-benzoylindoles were designed and synthesized as deaza analogues of our previously reported potent and selective HNE inhibitors with an indazole scaffold. The new compounds containing substituents and functions that were most active in the previous series were active in the micromolar r...

Szczegółowa specyfikacja

Zapisane w:
Opis bibliograficzny
Wydane w:Drug Dev Res
Główni autorzy: Crocetti, Letizia, Schepetkin, Igor A., Ciciani, Giovanna, Giovannoni, Maria Paola, Guerrini, Gabriella, Iacovone, Antonella, Khlebnikov, Andrei I., Kirpotina, Liliya N., Quinn, Mark T., Vergelli, Claudia
Format: Artigo
Język:Inglês
Wydane: 2016
Hasła przedmiotowe:
Dostęp online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5062748/
https://ncbi.nlm.nih.gov/pubmed/27474878
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/ddr.21323
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