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Bioactivation of Trimethoprim to Protein-Reactive Metabolites in Human Liver Microsomes

The formation of drug-protein adducts via metabolic activation and covalent binding may stimulate an immune response or may result in direct cell toxicity. Protein covalent binding is a potentially pivotal step in the development of idiosyncratic adverse drug reactions (IADRs). Trimethoprim (TMP)-su...

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Bibliografski detalji
Izdano u:Drug Metab Dispos
Glavni autori: Goldman, Jennifer L., Koen, Yakov M., Rogers, Steven A., Li, Kelin, Leeder, James S., Hanzlik, Robert P.
Format: Artigo
Jezik:Inglês
Izdano: The American Society for Pharmacology and Experimental Therapeutics 2016
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC5034695/
https://ncbi.nlm.nih.gov/pubmed/27457783
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.116.072041
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