Carregant...

A peptide of the RGS domain of GRK2 binds and inhibits Gα(q) to suppress pathological cardiac hypertrophy and dysfunction

G protein–coupled receptor (GPCR) kinases (GRKs) play a critical role in cardiac function by regulating GPCR activity. GRK2 suppresses GPCR signaling by phosphorylating and desensitizing active GPCRs, and through protein-protein interactions that uncouple GPCRs from their downstream effectors. Sever...

Descripció completa

Guardat en:
Dades bibliogràfiques
Publicat a:Sci Signal
Autors principals: Schumacher, Sarah M., Gao, Erhe, Cohen, Maya, Lieu, Melissa, Chuprun, J. Kurt, Koch, Walter J.
Format: Artigo
Idioma:Inglês
Publicat: 2016
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5015886/
https://ncbi.nlm.nih.gov/pubmed/27016525
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1126/scisignal.aae0549
Etiquetes: Afegir etiqueta
Sense etiquetes, Sigues el primer a etiquetar aquest registre!