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BCL2 inhibitors as anticancer drugs: a plethora of misleading BH3 mimetics

Anti-apoptotic BCL2 proteins play a major role in tumor cell survival. Hence, BCL2 inhibitors have been developed as direct inducers of apoptosis. ABT-199 (venetoclax) received breakthrough therapy designation from the FDA due to its apparent efficacy in CLL and AML. However, resistance to ABT-199 i...

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Publicat a:Mol Cancer Ther
Autors principals: Soderquist, Ryan S., Eastman, Alan
Format: Artigo
Idioma:Inglês
Publicat: 2016
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5010924/
https://ncbi.nlm.nih.gov/pubmed/27535975
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1158/1535-7163.MCT-16-0031
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