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Screening Identifies Thimerosal as a Selective Inhibitor of Endoplasmic Reticulum Aminopeptidase 1

[Image: see text] We employed virtual screening followed by in vitro evaluation to discover novel inhibitors of ER aminopeptidase 1, an important enzyme for the human adaptive immune response that has emerged as an attractive target for cancer immunotherapy and the control of autoimmunity. Screening...

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Опубликовано в: :ACS Med Chem Lett
Главные авторы: Stamogiannos, Athanasios, Papakyriakou, Athanasios, Mauvais, Francois-Xavier, van Endert, Peter, Stratikos, Efstratios
Формат: Artigo
Язык:Inglês
Опубликовано: American Chemical Society 2016
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC4948014/
https://ncbi.nlm.nih.gov/pubmed/27437077
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.6b00084
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