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Screening Identifies Thimerosal as a Selective Inhibitor of Endoplasmic Reticulum Aminopeptidase 1

[Image: see text] We employed virtual screening followed by in vitro evaluation to discover novel inhibitors of ER aminopeptidase 1, an important enzyme for the human adaptive immune response that has emerged as an attractive target for cancer immunotherapy and the control of autoimmunity. Screening...

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Detalles Bibliográficos
Publicado en:ACS Med Chem Lett
Main Authors: Stamogiannos, Athanasios, Papakyriakou, Athanasios, Mauvais, Francois-Xavier, van Endert, Peter, Stratikos, Efstratios
Formato: Artigo
Idioma:Inglês
Publicado: American Chemical Society 2016
Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC4948014/
https://ncbi.nlm.nih.gov/pubmed/27437077
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.6b00084
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