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Conversion of a single polypharmacological agent into selective bivalent inhibitors of intracellular kinase activity

Loss-of-function studies are valuable for elucidating kinase function and the validation of new drug targets. While genetic techniques, such as RNAi and genetic knockouts, are highly specific and easy to implement, in many cases post-translational perturbation of kinase activity, specifically pharma...

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Dades bibliogràfiques
Publicat a:ACS Chem Biol
Autors principals: Gower, Carrie M., Thomas, Jason R., Harrington, Edmund, Murphy, Jason, Chang, Matthew E. K., Cornella-Taracido, Ivan, Jain, Rishi K., Schirle, Markus, Maly, Dustin J.
Format: Artigo
Idioma:Inglês
Publicat: 2015
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4943861/
https://ncbi.nlm.nih.gov/pubmed/26505072
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschembio.5b00847
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