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Rational design and validation of a vanilloid-sensitive TRPV2 ion channel

Vanilloids activation of TRPV1 represents an excellent model system of ligand-gated ion channels. Recent studies using cryo-electron microcopy (cryo-EM), computational analysis, and functional quantification revealed the location of capsaicin-binding site and critical residues mediating ligand-bindi...

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Dettagli Bibliografici
Pubblicato in:Proc Natl Acad Sci U S A
Autori principali: Yang, Fan, Vu, Simon, Yarov-Yarovoy, Vladimir, Zheng, Jie
Natura: Artigo
Lingua:Inglês
Pubblicazione: National Academy of Sciences 2016
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4932969/
https://ncbi.nlm.nih.gov/pubmed/27298359
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1604180113
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