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Rationally Repurposing Ruxolitinib (Jakafi(®)) as a Solid Tumor Therapeutic

We determined whether the approved myelofibrosis drug ruxolitinib (Jakafi(®)), an inhibitor of Janus kinases 1/2 (JAK1 and JAK2), could be repurposed as an anti-cancer agent for solid tumors. Ruxolitinib synergistically interacted with dual ERBB1/2/4 inhibitors to kill breast as well as lung, ovaria...

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Detaylı Bibliyografya
Yayımlandı:Front Oncol
Asıl Yazarlar: Tavallai, Mehrad, Booth, Laurence, Roberts, Jane L., Poklepovic, Andrew, Dent, Paul
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: Frontiers Media S.A. 2016
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC4904019/
https://ncbi.nlm.nih.gov/pubmed/27379204
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3389/fonc.2016.00142
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