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An evaluation of Minor Groove Binders as anti-Trypanosoma brucei brucei therapeutics

A series of 32 structurally diverse MGBs, derived from the natural product distamycin, was evaluated for activity against Trypanosoma brucei brucei. Four compounds have been found to possess significant activity, in the nanomolar range, and represent hits for further optimisation towards novel treat...

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Detalhes bibliográficos
Publicado no:Eur J Med Chem
Main Authors: Scott, Fraser J., Khalaf, Abedawn I., Giordani, Federica, Wong, Pui Ee, Duffy, Sandra, Barrett, Michael, Avery, Vicky M., Suckling, Colin J.
Formato: Artigo
Idioma:Inglês
Publicado em: Editions Scientifiques Elsevier 2016
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4872591/
https://ncbi.nlm.nih.gov/pubmed/27060763
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ejmech.2016.03.064
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