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Pharmacologic efficacy of PU.1 inhibition by heterocyclic dications: a mechanistic analysis

Heterocyclic dications are receiving increasing attention as targeted inhibitors of transcription factors. While many dications act as purely competitive inhibitors, some fail to displace protein efficiently at drug concentrations expected to saturate their DNA target. To achieve a mechanistic under...

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Detalles Bibliográficos
Publicado en:Nucleic Acids Res
Main Authors: Stephens, Dominique C., Kim, Hye Mi, Kumar, Arvind, Farahat, Abdelbasset A., Boykin, David W., K. Poon, Gregory M.
Formato: Artigo
Idioma:Inglês
Publicado: Oxford University Press 2016
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC4872103/
https://ncbi.nlm.nih.gov/pubmed/27079976
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/nar/gkw229
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