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Design, synthesis, and kinetic analysis of potent protein N-terminal methyltransferase 1 inhibitors()

The protein N-terminal methyltransferase 1 (NTMT1) methylates the α-N-terminal amines of proteins. NTMT1 is upregulated in a variety of cancers and knockdown of NTMT1 results in cell mitotic defects. Therefore, NTMT1 inhibitors could be potential anticancer therapeutics. This study describes the des...

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Publicado en:Org Biomol Chem
Autores principales: Zhang, Gang, Richardson, Stacie Lynn, Mao, Yunfei, Huang, Rong
Formato: Artigo
Lenguaje:Inglês
Publicado: 2015
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC4857722/
https://ncbi.nlm.nih.gov/pubmed/25712161
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c5ob00120j
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