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Mechanism of Action Studies of Lomaiviticin A and the Monomeric Lomaiviticin Aglycon. Selective and Potent Activity Toward DNA Double-Strand Break Repair-Deficient Cell Lines

(−)-Lomaiviticin A (1) and the monomeric lomaiviticin aglycon [aka: (−)-MK7-206, (3)] are cytotoxic agents that induce double-strand breaks (DSBs) in DNA. Here we elucidate the cellular responses to these agents and identify synthetic lethal interactions with specific DNA repair factors. Toward this...

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Detalles Bibliográficos
Publicado en:J Am Chem Soc
Main Authors: Colis, Laureen C., Hegan, Denise C., Kaneko, Miho, Glazer, Peter M., Herzon, Seth B.
Formato: Artigo
Idioma:Inglês
Publicado: 2015
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC4845730/
https://ncbi.nlm.nih.gov/pubmed/25849366
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ja513117p
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