Caricamento...

Analgesia and unwanted benzodiazepine effects in point-mutated mice expressing only one benzodiazepine-sensitive GABA(A) receptor subtype

Agonists at the benzodiazepine-binding site of GABA(A) receptors (BDZs) enhance synaptic inhibition through four subtypes (α1, α2, α3 and α5) of GABA(A) receptors (GABA(A)R). When applied to the spinal cord, they alleviate pathological pain; however, insufficient efficacy after systemic administrati...

Descrizione completa

Salvato in:
Dettagli Bibliografici
Pubblicato in:Nat Commun
Autori principali: Ralvenius, William T., Benke, Dietmar, Acuña, Mario A., Rudolph, Uwe, Zeilhofer, Hanns Ulrich
Natura: Artigo
Lingua:Inglês
Pubblicazione: Nature Publishing Group 2015
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4829939/
https://ncbi.nlm.nih.gov/pubmed/25865415
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/ncomms7803
Tags: Aggiungi Tag
Nessun Tag, puoi essere il primo ad aggiungerne! !