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The anti-tumour agent lonidamine is a potent inhibitor of the mitochondrial pyruvate carrier and plasma membrane monocarboxylate transporters

Lonidamine (LND) is an anti-tumour drug particularly effective at selectively sensitising tumours to chemotherapy, hyperthermia and radiotherapy, although its precise mode of action remains unclear. It has been reported to perturb the bioenergetics of cells by inhibiting glycolysis and mitochondrial...

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Bibliographic Details
Published in:Biochem J
Main Authors: Nancolas, Bethany, Guo, Lili, Zhou, Rong, Nath, Kavindra, Nelson, David S., Leeper, Dennis B., Blair, Ian A., Glickson, Jerry D., Halestrap, Andrew P.
Format: Artigo
Language:Inglês
Published: 2016
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Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC4814305/
https://ncbi.nlm.nih.gov/pubmed/26831515
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1042/BJ20151120
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