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G Protein-Coupled Receptor Biased Agonism

G protein-coupled receptors (GPCR) are the largest family of targets for current therapeutics. The classic model of their activation was binary, where agonist binding induced an active conformation and subsequent downstream signaling. Subsequently, the revised concept of biased agonism emerged, wher...

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Detalles Bibliográficos
Publicado en:J Cardiovasc Pharmacol
Autores principales: Hodavance, Sima Y., Gareri, Clarice, Torok, Rachel D., Rockman, Howard A.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2016
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC4783281/
https://ncbi.nlm.nih.gov/pubmed/26751266
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1097/FJC.0000000000000356
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