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Uncoupling Catalytic and Binding Functions in the cAMP-Dependent Protein Kinase A

The canonical function of kinases is to transfer a phosphoryl group to substrates, initiating a signaling cascade; while their non-canonical role is to bind other kinases or substrates, acting as scaffolds, competitors, and signal integrators. Here, we show how to uncouple kinases dual function by t...

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發表在:Structure
Main Authors: Kim, Jonggul, Li, Geoffrey, Walters, Michael A., Taylor, Susan S., Veglia, Gianluigi
格式: Artigo
語言:Inglês
出版: 2016
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在線閱讀:https://ncbi.nlm.nih.gov/pmc/articles/PMC4775281/
https://ncbi.nlm.nih.gov/pubmed/26833386
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.str.2015.11.016
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