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A clickable psoralen to directly quantify DNA interstrand crosslinking and repair

DNA interstrand crosslinks (ICLs) represent physical obstacles to advancing replication forks and transcription complexes. A range of ICL-inducing agents have successfully been incorporated into cancer therapeutics. While studies have adopted UVA-activated psoralens as model ICL-inducing agents for...

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Detalles Bibliográficos
Publicado en:Bioorg Med Chem
Autores principales: Evison, Benjamin J., Actis, Marcelo L., Fujii, Naoaki
Formato: Artigo
Lenguaje:Inglês
Publicado: 2016
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC4762217/
https://ncbi.nlm.nih.gov/pubmed/26833244
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2016.01.032
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