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Kinase inhibitor profiling reveals unexpected opportunities to inhibit disease-associated mutant kinases

Small-molecule kinase inhibitors have typically been designed to inhibit wild-type kinases rather than the mutant forms that frequently arise in diseases such as cancer. Mutations can have serious clinical implications by increasing kinase catalytic activity or conferring therapeutic resistance. To...

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Detalhes bibliográficos
Publicado no:Cell Rep
Main Authors: Duong-Ly, Krisna C., Devarajan, Karthik, Liang, Shuguang, Horiuchi, Kurumi Y., Wang, Yuren, Ma, Haiching, Peterson, Jeffrey R.
Formato: Artigo
Idioma:Inglês
Publicado em: 2016
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4740242/
https://ncbi.nlm.nih.gov/pubmed/26776524
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.celrep.2015.12.080
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