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Covalent targeting of acquired cysteines in cancer

The thiolate side chain of cysteine has a unique functionality that drug hunters and chemical biologists have begun to exploit. For example, targeting cysteine residues in the ATP-binding pockets of kinases with thiol-reactive molecules has afforded increased selectivity and potency to drugs like im...

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Foilsithe in:Curr Opin Chem Biol
Main Authors: Visscher, Marieke, Arkin, Michelle R., Dansen, Tobias B.
Formáid: Artigo
Teanga:Inglês
Foilsithe: 2015
Ábhair:
Rochtain Ar Líne:https://ncbi.nlm.nih.gov/pmc/articles/PMC4731306/
https://ncbi.nlm.nih.gov/pubmed/26629855
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.cbpa.2015.11.004
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