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Macromolecular Modelling and Docking Simulations for the Discovery of Selective GPER Ligands

Estrogens influence multiple physiological processes and are implicated in many diseases as well. Cellular responses to estrogens are mainly mediated by the estrogen receptors (ER)α and ERβ, which act as ligand-activated transcription factors. Recently, a member of the G protein-coupled receptor (GP...

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Detalhes bibliográficos
Publicado no:AAPS J
Main Authors: Rosano, Camillo, Ponassi, Marco, Santolla, Maria Francesca, Pisano, Assunta, Felli, Lamberto, Vivacqua, Adele, Maggiolini, Marcello, Lappano, Rosamaria
Formato: Artigo
Idioma:Inglês
Publicado em: Springer US 2015
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4706286/
https://ncbi.nlm.nih.gov/pubmed/26573009
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1208/s12248-015-9844-3
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