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Design, Synthesis, Biological Evaluation and X-ray Structural Studies of HIV-1 Protease Inhibitors Containing Substituted Fused-Tetrahydropyranyl Tetrahydrofuran as P2-Ligands

Design, synthesis, biological and X-ray crystallographic studies of a series of potent HIV-1 protease inhibitors are described. Various polar functionalities have been incorporated on the tetrahydropyranyl-tetrahydrofuran-derived P2 ligand to interact with the backbone atoms in the S2 subsite. The m...

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Detalhes bibliográficos
Publicado no:Org Biomol Chem
Main Authors: Ghosh, Arun K., Martyr, Cuthbert D., Kassekert, Luke A., Nyalapatla, Prasanth R., Steffey, Melinda, Agniswamy, Johnson, Wang, Yuan-Fang, Weber, Irene T., Amano, Masayuki, Mitsuya, Hiroaki
Formato: Artigo
Idioma:Inglês
Publicado em: 2015
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4666783/
https://ncbi.nlm.nih.gov/pubmed/26462551
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c5ob01930c
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