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Highly Potent HIV-1 Protease Inhibitors with Novel Tricyclic P2-ligands: Design, Synthesis, and Protein-ligand X-Ray Studies

The design, synthesis, and biological evaluation of a series of HIV-1 protease inhibitors incorporating stereochemically defined fused tricyclic P2-ligands are described. Various substituent effects were investigated in order to maximize the ligand-binding site interactions in the protease active si...

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Detalhes bibliográficos
Main Authors: Ghosh, Arun K., Parham, Garth L., Martyr, Cuthbert D., Nyalapatla, Prasanth R., Osswald, Heather L., Agniswamy, Johnson, Wang, Yuan-Fang, Amano, Masayuki, Weber, Irene T., Mitsuya, Hiroaki
Formato: Artigo
Idioma:Inglês
Publicado em: 2013
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3800042/
https://ncbi.nlm.nih.gov/pubmed/23947685
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm400768f
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