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Total Synthesis and Absolute Stereochemistry of the Proteasome Inhibitors Cystargolides A and B

The absolute stereochemistry of the cystargolides was determined by total synthesis. Evaluation of synthetic cystargolides and derivatives showed that the natural (2S,3R) stereochemistry is essential for activity. Moreover, benzyl esters (−)-10 and (−)-15 were found to be about 100 times more potent...

पूर्ण विवरण

में बचाया:
ग्रंथसूची विवरण
में प्रकाशित:Org Biomol Chem
मुख्य लेखकों: Tello-Aburto, Rodolfo, Hallada, Liam P., Niroula, Doleshwar, Rogelj, Snezna
स्वरूप: Artigo
भाषा:Inglês
प्रकाशित: 2015
विषय:
ऑनलाइन पहुंच:https://ncbi.nlm.nih.gov/pmc/articles/PMC4629797/
https://ncbi.nlm.nih.gov/pubmed/26400369
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c5ob01821h
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