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Design, Synthesis, and Evaluation of Cystargolide-based β-lactones as Potent Proteasome Inhibitors

The peptidic β-lactone proteasome inhibitors (PIs) cystargolides A and B were used to conduct structure-activity relationship (SAR) studies in order to assess their anticancer potential. A total of 24 different analogs were designed, synthesized and evaluated for proteasome inhibition, for cytotoxic...

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Detalhes bibliográficos
Publicado no:Eur J Med Chem
Main Authors: Niroula, Doleshwar, Hallada, Liam P, Le Chapelain, Camille, Ganegamage, Susantha K, Dotson, Devon, Rogelj, Snezna, Groll, Michael, Tello-Aburto, Rodolfo
Formato: Artigo
Idioma:Inglês
Publicado em: 2018
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6168434/
https://ncbi.nlm.nih.gov/pubmed/30165344
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ejmech.2018.08.052
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