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An Unprecedented Dual Antagonist and Agonist of Human Transglutaminase 2

Transglutaminase 2 (TG2) is a ubiquitously expressed, Ca(2+)-activated extracellular enzyme in mammals that is maintained in a catalytically dormant state by multiple mechanisms. Although its precise physiological role in the extracellular matrix remains unclear, aberrantly up-regulated TG2 activity...

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Dettagli Bibliografici
Pubblicato in:Bioorg Med Chem Lett
Autori principali: Yi, Michael C, Palanski, Brad A, Quintero, Steven A, Plugis, Nicholas M, Khosla, Chaitan
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2015
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4607565/
https://ncbi.nlm.nih.gov/pubmed/26004580
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2015.05.006
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