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Pentafluorosulfanyl-containing flufenamic acid analogs: Syntheses, properties and biological activities

Pentafluorosulfanyl-containing analogs of flufenamic acid have been synthesized in high yields. Computationally, pK(a), logP and logD values have been determined. Initial bioactivity studies reveal effects as ion channel modulators and inhibitory activities on aldo-keto reductase 1C3 (AKR1C3) as wel...

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Bibliografiske detaljer
Udgivet i:Bioorg Med Chem Lett
Main Authors: Hendriks, Christine M. M., Penning, Trevor M., Zang, Tianzhu, Wiemuth, Dominik, Gründer, Stefan, Sanhueza, Italo A., Schoenebeck, Franziska, Bolm, Carsten
Format: Artigo
Sprog:Inglês
Udgivet: 2015
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC4599580/
https://ncbi.nlm.nih.gov/pubmed/26372652
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2015.09.012
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