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Synthesis and biological evaluation of the first pentafluorosulfanyl analogs of mefloquine

Two novel SF(5) analogs of the antimalarial agent mefloquine were synthesized in 5 steps and 10–23% overall yields and found to have improved activity and selectivity against malaria parasites. This work also represents the first report of SF(5)-substituted quinolines.

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Detalhes bibliográficos
Main Authors: Wipf, Peter, Mo, Tingting, Geib, Steven J., Caridha, Diana, Dow, Geoffrey S., Gerena, Lucia, Roncal, Norma, Milner, Erin E.
Formato: Artigo
Idioma:Inglês
Publicado em: 2009
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2929370/
https://ncbi.nlm.nih.gov/pubmed/19795052
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/b911483a
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