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Identification of non-peptidic cysteine reactive fragments as inhibitors of cysteine protease rhodesain

Rhodesain, the major cathepsin L-like cysteine protease in the protozoan Trypanosoma brucei rhodesiense, the causative agent of African sleeping sickness, is a well-validated drug target. In this work, we used a fragment-based approach to identify inhibitors of this cysteine protease, and identified...

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Detalhes bibliográficos
Publicado no:Bioorg Med Chem Lett
Main Authors: McShan, Danielle, Kathman, Stefan, Lowe, Brittiney, Xu, Ziyang, Zhan, Jennifer, Statsyuk, Alexander, Ogungbe, Ifedayo Victor
Formato: Artigo
Idioma:Inglês
Publicado em: 2015
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4592840/
https://ncbi.nlm.nih.gov/pubmed/26342866
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2015.08.074
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