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Rational Design of Orthogonal Multipolar Interactions with Fluorine in Protein–Ligand Complexes

[Image: see text] Multipolar interactions involving fluorine and the protein backbone have been frequently observed in protein–ligand complexes. Such fluorine–backbone interactions may substantially contribute to the high affinity of small molecule inhibitors. Here we found that introduction of trif...

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Detalhes bibliográficos
Publicado no:J Med Chem
Main Authors: Pollock, Jonathan, Borkin, Dmitry, Lund, George, Purohit, Trupta, Dyguda-Kazimierowicz, Edyta, Grembecka, Jolanta, Cierpicki, Tomasz
Formato: Artigo
Idioma:Inglês
Publicado em: American Chemical Society 2015
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4584387/
https://ncbi.nlm.nih.gov/pubmed/26288158
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.5b00975
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