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Pyridine-Substituted Desoxyritonavir Is a More Potent Inhibitor of Cytochrome P450 3A4 than Ritonavir

Utilization of the cytochrome P450 3A4 (CYP3A4) inhibitor ritonavir as a pharmacoenhancer for anti-HIV drugs revolutionized the treatment of HIV infection. However, owing to ritonavir-related complications, there is a need for development of new CYP3A4 inhibitors with improved pharmacochemical prope...

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Detalles Bibliográficos
Publicado en:J Med Chem
Autores principales: Sevrioukova, Irina F., Poulos, Thomas L.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2013
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC4534002/
https://ncbi.nlm.nih.gov/pubmed/23586711
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm400288z
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