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Combinatorial active-site variants confer sustained clavulanate resistance in BlaC β-lactamase from Mycobacterium tuberculosis

Bacterial resistance to β-lactam antibiotics is a global issue threatening the success of infectious disease treatments worldwide. Mycobacterium tuberculosis has been particularly resilient to β-lactam treatment, primarily due to the chromosomally encoded BlaC β-lactamase, a broad-spectrum hydrolase...

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Publicat a:Protein Sci
Autors principals: Egesborg, Philippe, Carlettini, Hélène, Volpato, Jordan P, Doucet, Nicolas
Format: Artigo
Idioma:Inglês
Publicat: Blackwell Publishing Ltd 2015
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4380984/
https://ncbi.nlm.nih.gov/pubmed/25492589
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/pro.2617
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