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New Inhibitor of 3-Phosphoinositide Dependent Protein Kinase-1 Identified from Virtual Screening

3-Phosphoinositide-dependent protein kinase-1 (PDK1) has been recognized as a promising anticancer target. Thus, it is interesting to identify new inhibitors of PDK1 for anticancer drug discovery. Through a combined use of virtual screening and wet experimental activity assays, we have identified a...

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Pubblicato in:Bioorg Med Chem Lett
Autori principali: Yang, Wenchao, AbdulHameed, Mohamed Diwan M., Hamza, Adel, Zhan, Chang-Guo
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2012
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4371734/
https://ncbi.nlm.nih.gov/pubmed/22266037
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2011.12.121
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