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Quantification of Histone H3 Lys27 Trimethylation (H3K27me3) by High-Throughput Microscopy Enables Cellular Large-Scale Screening for Small-Molecule EZH2 Inhibitors

EZH2 inhibition can decrease global histone H3 lysine 27 trimethylation (H3K27me3) and thereby reactivates silenced tumor suppressor genes. Inhibition of EZH2 is regarded as an option for therapeutic cancer intervention. To identify novel small-molecule (SMOL) inhibitors of EZH2 in drug discovery, t...

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Bibliografiska uppgifter
I publikationen:J Biomol Screen
Huvudupphovsmän: Luense, Svenja, Denner, Philip, Fernández-Montalván, Amaury, Hartung, Ingo, Husemann, Manfred, Stresemann, Carlo, Prechtl, Stefan
Materialtyp: Artigo
Språk:Inglês
Publicerad: SAGE Publications 2015
Ämnen:
Länkar:https://ncbi.nlm.nih.gov/pmc/articles/PMC4361481/
https://ncbi.nlm.nih.gov/pubmed/25409661
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1177/1087057114559668
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