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Metabolism-Directed Structure Optimization of Benzimidazole-Based Francisella tularensis Enoyl-Reductase (FabI) Inhibitors

FabI is a potential antibiotic target against Francisella tularensis, which has been classified as a Category A biowarfare agent of high risk to public health. Our previous work demonstrated that N-benzyl benzimidazole compounds possess promising FabI inhibitory activity, but their druggability prop...

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Kaydedildi:
Detaylı Bibliyografya
Yayımlandı:Xenobiotica
Asıl Yazarlar: Zhang, Yan-Yan, Liu, Yong, Mehboob, Shahila, Song, Jin-Hua, Boci, Teuta, Johnson, Michael E., Ghosh, Arun K., Jeong, Hyunyoung
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: 2013
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC4355941/
https://ncbi.nlm.nih.gov/pubmed/24171690
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3109/00498254.2013.850553
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