Loading...

Mechanism of initiation of aggregation of p53 revealed by Φ-value analysis

Many oncogenic mutations inactivate the tumor suppressor p53 by destabilizing it, leading to its rapid aggregation. Small molecule drugs are being developed to stabilize such mutants. The kinetics of aggregation of p53 is deceptively simple. The initial steps in the micromolar concentration range fo...

Full description

Saved in:
Bibliographic Details
Published in:Proc Natl Acad Sci U S A
Main Authors: Wang, GuoZhen, Fersht, Alan R.
Format: Artigo
Language:Inglês
Published: National Academy of Sciences 2015
Subjects:
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC4345617/
https://ncbi.nlm.nih.gov/pubmed/25675526
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1500243112
Tags: Add Tag
No Tags, Be the first to tag this record!