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The Extracellular Loop 2 (ECL2) of the Human Histamine H(4) Receptor Substantially Contributes to Ligand Binding and Constitutive Activity

In contrast to the corresponding mouse and rat orthologs, the human histamine H(4) receptor (hH(4)R) shows extraordinarily high constitutive activity. In the extracellular loop (ECL), replacement of F169 by V as in the mouse H(4)R significantly reduced constitutive activity. Stabilization of the ina...

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Publicado en:PLoS One
Main Authors: Wifling, David, Bernhardt, Günther, Dove, Stefan, Buschauer, Armin
Formato: Artigo
Idioma:Inglês
Publicado: Public Library of Science 2015
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC4309601/
https://ncbi.nlm.nih.gov/pubmed/25629160
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0117185
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