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DESIGN, SYNTHESIS, AND EVALUATION OF A FAMILY OF PROPARGYL PYRIDINYL ETHERS AS POTENTIAL CYTOCHROME P450 INHIBITORS

Cytochrome P450 enzymes are a superfamily of hemoproteins involved in the metabolism of endogenous and exogenous compounds including many drugs and environmental chemicals. In our previous research, we have determined that certain aryl and arylalkyl acetylenes act as inhibitors of these enzymes. Her...

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Publicado en:J Undergrad Chem Res
Autores principales: Foroozesh, Maryam, Jiang, Quan, Sridhar, Jayalakshmi, Liu, Jiawang, Minaruzzaman, Dotson, Brandan, McClain, Erika
Formato: Artigo
Lenguaje:Inglês
Publicado: 2013
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC4275839/
https://ncbi.nlm.nih.gov/pubmed/25544835
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