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DESIGN, SYNTHESIS, AND EVALUATION OF A FAMILY OF PROPARGYL PYRIDINYL ETHERS AS POTENTIAL CYTOCHROME P450 INHIBITORS

Cytochrome P450 enzymes are a superfamily of hemoproteins involved in the metabolism of endogenous and exogenous compounds including many drugs and environmental chemicals. In our previous research, we have determined that certain aryl and arylalkyl acetylenes act as inhibitors of these enzymes. Her...

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Publicat a:J Undergrad Chem Res
Autors principals: Foroozesh, Maryam, Jiang, Quan, Sridhar, Jayalakshmi, Liu, Jiawang, Minaruzzaman, Dotson, Brandan, McClain, Erika
Format: Artigo
Idioma:Inglês
Publicat: 2013
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4275839/
https://ncbi.nlm.nih.gov/pubmed/25544835
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