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Characterization of [(3)H]LS-3-134, a Novel Arylamide Phenylpiperazine D3 Dopamine Receptor Selective Radioligand

LS-3-134 is a substituted N-phenylpiperazine derivative that has been reported to exhibit a) high-affinity binding (Ki value 0.2 nM) at human D3 dopamine receptors, b) >100-fold D3 vs. D2 dopamine receptor subtype binding selectivity and c) low-affinity binding (Ki values >5,000 nM) at sigma 1...

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Bibliografski detalji
Izdano u:J Neurochem
Glavni autori: Rangel-Barajas, Claudia, Malik, Maninder, Taylor, Michelle, Neve, Kim A., Mach, Robert H., Luedtke, Robert R.
Format: Artigo
Jezik:Inglês
Izdano: 2014
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC4222986/
https://ncbi.nlm.nih.gov/pubmed/25041389
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/jnc.12825
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