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Substantial Non-Electrostatic Forces Are Needed To Induce Allosteric Disruption of Thrombin’s Active Site Through Exosite 2

Sulfated beta-O4 lignin (SbO4L), a non-saccharide glycosaminoglycan mimetic, was recently disclosed as a novel exosite 2-directed thrombin inhibitor with capability of mimicking sulfated tyrosine sequences of glycoprotein Ibα resulting in dual anticoagulant and antiplatelet activities. SbO4L engages...

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Detalhes bibliográficos
Main Authors: Mehta, Akul Y., Desai, Umesh R.
Formato: Artigo
Idioma:Inglês
Publicado em: 2014
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4179500/
https://ncbi.nlm.nih.gov/pubmed/25201728
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bbrc.2014.09.003
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