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Designing Allosteric Regulators of Thrombin. Exosite 2 Features Multiple Sub-Sites That Can Be Targeted By Sulfated Small Molecules for Inducing Inhibition

We recently designed a group of novel exosite 2-directed, sulfated, small, allosteric inhibitors of thrombin. To develop more potent inhibitors, monosulfated benzofuran tri- and tetrameric homologs of the parent designed dimers were synthesized in 7–8 steps and found to exhibit a wide range of poten...

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Detalhes bibliográficos
Main Authors: Sidhu, Preetpal Singh, Abdel Aziz, May H., Sarkar, Aurijit, Mehta, Akul Y., Zhou, Qibing, Desai, Umesh R.
Formato: Artigo
Idioma:Inglês
Publicado em: 2013
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3717983/
https://ncbi.nlm.nih.gov/pubmed/23718540
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm400369q
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