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Influence of Macrocyclization on Allosteric, Juxtamembrane-Derived, Stapled Peptide Inhibitors of the Epidermal Growth Factor Receptor (EGFR)

[Image: see text] The hydrocarbon-stapled peptide E1(S) allosterically inhibits the kinase activity of the epidermal growth factor receptor (EGFR) by blocking a distant but essential protein–protein interaction: a coiled coil formed from the juxtamembrane segment (JM) of each member of the dimeric p...

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Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: Sinclair, Julie K.-L., Schepartz, Alanna
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: American Chemical Society 2014
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC4168776/
https://ncbi.nlm.nih.gov/pubmed/25207804
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ol502426b
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